找到约 30 条 “Dopamine Receptor” 相关结果 (用时 0.074 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M2372 | Alizapride hydrochloride | 盐酸阿立必利 | Dopamine Receptor |
Alizapride HCl 是一种 dopamine receptor 拮抗剂,用于恶心和呕吐的治疗。 | |||
M2494 | Cariprazine hydrochloride | 盐酸卡利拉嗪;卡利拉嗪盐酸盐 | Dopamine Receptor |
RGH-188 HCl | |||
Cariprazine hydrochloride是一种dopamine D3-receptor(多巴胺D3受体)部分激动剂,作用于dopamine D3和D2受体具有高度选择性和亲和力,pKi分别为10.07, 9.16和9.31。 | |||
M2886 | Nomifensine Maleate | 诺米芬新马来酸盐 | Dopamine Receptor |
(±)-Nomifensine maleat | |||
Nomifensine is a dopamine reuptake inhibitor that increases the amount of synaptic dopamine available to receptors by blocking dopamine's re-uptake transporter. | |||
M2945 | Pimozide | 匹莫奇特;哌咪清 | Dopamine Receptor |
R6238 | |||
Pimozide 是 dopamine receptor 的拮抗剂,对 dopamine D2,D3 和 D1 受体的 Ki 值分别为 1.4 nM,2.5 nM 和 588 nM,同时对 α1-adrenoceptor 也有较高亲和性,Ki 值为 39 nM;Pimozide 也是 STAT3 和 STAT5 的抑制剂,哌咪清可通过诱导mTORC1去磷酸化和失活,在胶质母细胞瘤细胞系(LN-229、MZ-54、GOS-3和U343)中触发ADCD。 | |||
M3320 | Quetiapine Fumarate | 富马酸喹硫平 | 5-HT Receptor |
Quetiapine hemifumarate | |||
Quetiapine Fumarate是一种 5-HT 受体激动剂,对人 5-HT1A 的 pEC50 值为 4.77。Quetiapine hemifumarate 是多巴胺受体 (dopamine receptor) 拮抗剂,对人 D2 的 pIC50 值为 6.33。 | |||
M3675 | Rotigotine | 罗替戈汀 | Dopamine Receptor |
N-0923 | |||
Rotigotine (N-0437; N-0923) 是 dopamine receptor 激动剂,是 5-HT1A receptor 的部分激动剂,以及 α2B-adrenergic receptor 的拮抗剂,Ki 值分别为 0.71 nM (dopamine D3 receptor),4-15 nM (D2,D5,D4 receptors),83 nM (dopamine D1 receptor)。 | |||
M3818 | Rotigotine Hydrochloride | 罗替戈汀盐酸盐 | Dopamine Receptor |
Rotigotine HCl;N-0923 Hydrochloride | |||
Rotigotine Hydrochloride (N-0923 Hydrochloride) 是 dopamine receptor 纯激动剂,是 5-HT1A receptor 的部分激动剂,以及 α2B-adrenergic receptor 的拮抗剂,Ki 值分别为 0.71 nM (dopamine D3 receptor),4-15 nM (D2,D5,D4 receptors),83 nM (dopamine D1 receptor)。 | |||
M1574 | Iloperidone | 伊潘立酮 | 5-HT Receptor |
HP873 | |||
Iloperidone是一种dopamine (D2)/serotonin (5-HT2) receptor抑制剂,用于研究精神分裂症。 | |||
M1565 | Quetiapine sulfoxide | 喹硫平硫氧化物/喹硫平亚砜 | 5-HT Receptor |
Quetiapine sulfoxide; Quetiapine S-oxide | |||
Quetiapine sulfoxide是一种 5-HT 受体激动剂,对人 5-HT1A 的 pEC50 值为 4.77。Quetiapine hemifumarate 是多巴胺受体 (dopamine receptor) 拮抗剂,对人 D2 的 pIC50 值为 6.33。 | |||
M1564 | Quetiapine Sulfone | 喹硫平砜 | 5-HT Receptor |
Quetiapine Sulfone是一种 5-HT 受体激动剂,对人 5-HT1A 的 pEC50 值为 4.77。Quetiapine hemifumarate 是多巴胺受体 (dopamine receptor) 拮抗剂,对人 D2 的 pIC50 值为 6.33。 | |||
M4887 | Pardoprunox Hydrochloride | 盐酸帕多芦诺 | 5-HT Receptor |
SLV-308 | |||
Pardoprunox hydrochloride (DU-126891, SME-308)是一种有效的部分 dopamine D2 receptor 的激动剂,对应的pEC50值为8.0,也是诱导 [35S]GTPγS binding 的部分激动剂,对应的pEC50值为9.2,和 serotonin 5-HT1A receptor 的激动剂,pEC50值为6.3。 | |||
M5350 | Octopamine hydrochloride | (±)-章胺盐酸盐 | Dopamine Receptor |
(±)-p-Octopamine hydrochloride | |||
(±)-Octopamine HCl 是一种生命必需的一元胺,结构上与去甲肾上腺素相关,是一种内源性多巴胺D-1受体(Dopamine Receptor)阻断剂,在无脊椎动物中作为一种神经激素,神经调节物质以及神经递质。 | |||
M5590 | Dopamine HCl | 盐酸多巴胺 | Dopamine Receptor |
ASL279; Dopamine hydrochloride | |||
Dopamine HCl 是一种广泛存在于各种动物的儿茶酚胺类神经递质,是多巴胺D1-5受体(Dopamine Receptor)激动剂。Dopamine hydrochloride (ASL279) 通过 D2 多巴胺受体 (D2 dopamine receptor) 来诱导 VEGFR2 的内吞作用。 | |||
M5642 | Fenoldopam mesylate | 甲磺酸非诺多泮 | Dopamine Receptor |
KF 82526 (mesylate), Fenoldopam methanesulfonate, Corlopam mesylate | |||
Fenoldopam是一种选择性的多巴胺受体(dopamine-1 receptor)激动剂。 | |||
M5984 | Sulpiride | 舒必利 | Dopamine Receptor |
Dolmatil, Dobren, Sulpyrid, Aiglonyl, Dogmatil | |||
Sulpiride是一种多巴胺D2受体(Dopamine Receptor)拮抗剂。 | |||
M6064 | Ziprasidone HCl | 盐酸齐拉西酮 | 5-HT Receptor |
CP-88059 | |||
Ziprasidone HCl 是一类有效的Dopamine 和 Serotonin (5-HT) Receptor的拮抗剂,可用于精神分裂症以及双向性障碍的相关研究。 | |||
M6950 | Mesulergine hydrochloride | Mesulergine hydrochloride | Others |
Mesulergine hydrochloride is a 5-HT 2A and 5-HT 2C antagonist. Also dopamine receptor partial agonist. | |||
M7213 | Roxindole hydrochloride | Roxindole hydrochloride | Others |
Roxindole hydrochloride is a dopamine D 2 autoreceptor agonist. Also has affinity for D 3, D 4, 5-HT 1A receptors and the 5-HT transporter. | |||
M7656 | BP897 | BP897 | Others |
Partially selective D3 dopamine receptor agonist. | |||
M7697 | Chlorprothixene hydrochloride | 盐酸氯普噻吨 | Others |
D2 dopamine receptor antagonist; blocks a subset of GABAA receptors in rat cortex that is also blocked by clozapine; thioxanthine antipsychotic. | |||
M7739 | (+)-Butaclamol hydrochloride | (+)-Butaclamol hydrochloride | Others |
(+)-Butaclamol is a dopamine receptor antagonist; active enantiomer. | |||
M7803 | FAUC 213 | FAUC 213 | Others |
Highly selective D4 dopamine receptor full antagonist. | |||
M7830 | Halopemide | 卤培米特 | Others |
Halopemide is a dopamine receptor antagonist and a phospholipase D2 inhibitor. | |||
M7883 | L-741,626 | L-741,626 | Others |
Selective D2 dopamine receptor antagonist. | |||
M7977 | Octoclothepin maleate salt | Octoclothepin maleate salt | Others |
Octoclothepin maleate salt is a D2 dopamine receptor antagonist; 5-HT2 serotonin receptor antagonist. | |||
M8003 | (+)-PD 128,907 hydrochloride | (+)-PD 128,907 hydrochloride | Others |
Selective D3 dopamine receptor agonist. | |||
M8005 | PD 168,077 maleate salt | PD 168,077 maleate salt | Others |
Selective D4 dopamine receptor agonist. | |||
M8009 | Pipamperone dihydrochloride | Pipamperone dihydrochloride | Others |
D2 dopamine receptor antagonist; 5-HT2 serotonin receptor antagonist; antipsychotic. | |||
M8024 | Propionylpromazine hydrochloride | 盐酸丙酰丙嗪 | Others |
Phenothiazine antipsychotic; D2 dopamine receptor antagonist. | |||
M8039 | CP-226269 | CP-226269 | Others |
CP-226269 is a D4 dopamine receptor agonist with EC50 of 32 nM. |
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